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Wynne Aherne Selected Research

VER-50589

4/2007Inhibition of the heat shock protein 90 molecular chaperone in vitro and in vivo by novel, synthetic, potent resorcinylic pyrazole/isoxazole amide analogues.

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Wynne Aherne Research Topics

Disease

30Neoplasms (Cancer)
09/2012 - 09/2003
3Colonic Neoplasms (Colon Cancer)
12/2011 - 04/2007
3Melanoma (Melanoma, Malignant)
03/2011 - 03/2007
3Carcinoma (Carcinomatosis)
04/2008 - 04/2007
2Glioblastoma (Glioblastoma Multiforme)
02/2011 - 01/2011
2Hypoxia (Hypoxemia)
04/2008 - 06/2005
2Neoplasm Metastasis (Metastasis)
04/2008 - 06/2005
1Prostatic Neoplasms (Prostate Cancer)
03/2011
1Chondrosarcoma
03/2011
1Kidney Neoplasms (Kidney Cancer)
03/2011
1Breast Neoplasms (Breast Cancer)
02/2011
1Atrial Fibrillation
10/2008
1Fatigue
10/2008
1Hyperbilirubinemia
10/2008
1Lymphatic Metastasis
04/2008
1Squamous Cell Carcinoma (Epidermoid Carcinoma)
07/2007
1Ovarian Neoplasms (Ovarian Cancer)
04/2007
1Osteosarcoma (Osteogenic Sarcoma)
06/2005

Drug/Important Bio-Agent (IBA)

12Pharmaceutical PreparationsIBA
02/2011 - 04/2004
9Proteins (Proteins, Gene)FDA Link
03/2011 - 06/2004
8Heat-Shock Proteins (Heat-Shock Protein)IBA
12/2011 - 06/2005
3Histones (Histone)IBA
11/2010 - 05/2004
3Molecular Chaperones (Chaperone, Molecular)IBA
03/2010 - 06/2005
2EnzymesIBA
09/2012 - 05/2004
2Phosphotransferases (Kinase)IBA
01/2012 - 09/2010
2AcidsIBA
12/2011 - 09/2010
2monorden (radicicol)IBA
12/2011 - 09/2010
2Biological ProductsIBA
12/2011 - 09/2010
2Biomarkers (Surrogate Marker)IBA
02/2011 - 06/2007
2Adenosine Triphosphatases (ATPase)IBA
03/2010 - 06/2004
2HSP72 Heat-Shock ProteinsIBA
03/2010 - 03/2007
2LAQ824IBA
10/2008 - 04/2008
2Histone Deacetylase InhibitorsIBA
10/2008 - 04/2008
25- (2,4- dihydroxy- 5- isopropylphenyl)- 4- (4- morpholin- 4- ylmethylphenyl)isoxazole- 3- carboxylic acid ethylamideIBA
04/2008 - 01/2008
2IsoxazolesIBA
04/2008 - 04/2007
2Phosphatidylinositol 3-Kinases (PI 3 Kinase)IBA
06/2007 - 10/2006
1ChromatinIBA
09/2012
1Macrocyclic LactamsIBA
12/2011
1LactonesIBA
12/2011
1NitrogenIBA
12/2011
117- (dimethylaminoethylamino)- 17- demethoxygeldanamycinIBA
03/2011
1Adenosine Triphosphate (ATP)IBA
03/2011
14- (4- chlorobenzyl)- 1- (7H- pyrrolo(2,3- d)pyrimidin- 4- yl)piperidin- 4- amineIBA
02/2011
1Angiogenesis InhibitorsIBA
01/2011
1Tissue Inhibitor of Metalloproteinase-1IBA
01/2011
1AminesIBA
11/2010
1Histone Deacetylases (Histone Deacetylase)IBA
11/2010
1beta CateninIBA
07/2010
1CreatinineIBA
10/2008
1Cyclin-Dependent Kinase 4IBA
04/2008
1Therapeutic UsesIBA
04/2008
1tris-O-tolyphosphine (TOTP)IBA
04/2008
1triphosphoric acid (triphosphate)IBA
04/2008
1NucleosidesIBA
04/2008
1Phosphates (Orthophosphate)IBA
04/2008
1Phosphorus (Red Phosphorus)IBA
04/2008
1Phosphorylcholine (Phosphocholine)IBA
04/2008
1VorinostatFDA Link
04/2008
1Phospholipids (Phosphatides)FDA LinkGeneric
04/2008
11- (6- ((3- methoxyestra- 1,3,5(10)- trien- 17- yl)amino)hexyl)- 1H- pyrrole- 2,5- dioneIBA
07/2007
1Epidermal Growth Factor (EGF)IBA
07/2007
1Glycogen Synthase (Synthase I)IBA
06/2007
1Phosphatidylinositols (Phosphatidylinositol)IBA
06/2007
1PhosphoproteinsIBA
06/2007
12- (4- morpholinyl)- 8- phenyl- 4H- 1- benzopyran- 4- oneIBA
06/2007
1VER-49009IBA
04/2007
1VER-50589IBA
04/2007
1tanespimycin (17AAG)IBA
04/2007
1HSP27 Heat-Shock ProteinsIBA
04/2007
1CCT018159IBA
03/2007
1Proto-Oncogene Proteins c-akt (Protein Kinase B)IBA
10/2006
1Deferoxamine (Desferal)FDA LinkGeneric
06/2005
1NSC-134754IBA
06/2005
1Intercellular Signaling Peptides and Proteins (Growth Factors)IBA
06/2005
1LuciferasesIBA
06/2005
1Aurora KinasesIBA
05/2004
1Histone MethyltransferasesIBA
05/2004
1CyclinsIBA
09/2003

Therapy/Procedure

2Therapeutics
01/2011 - 12/2006
1Castration
03/2011
1Aftercare (After-Treatment)
04/2008